SCHEMBL8666901

SCHEMBL8666901

Cn1cc(C(C(=O)O)C(F)(F)F)nc1-c1ccc(-c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.42
DHODH Q02127 2/20 0.38
CYP1A2 P05177 2/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
PKM P14618 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGS1 P23219 1/20 0.36
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
MMP1 P03956 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8666893 0.80 PTGS2 (0.39) PTGS2DHODHCYP1A2GAACYP2C9
SCHEMBL25147202 0.75 MC4R (0.42) PDE3BPDE3ANR1H2NR1H3
SCHEMBL8666707 0.75 COMT (0.42) PTGS2DHODHPDE3BPDE3AKMT2A
SCHEMBL6976337 0.69 HPGD (0.38) PDE3BPDE3ANR1H2NR1H3
SCHEMBL2278129 0.69 PDE3B (0.37) CYP1A2GAAPDE3BPDE3ANR1H2
SCHEMBL2224580 0.69 TAAR1 (0.42) PDE3BPDE3AKMT2ANR1H2NR1H3
SCHEMBL8666896 0.68 KDM4E (0.44) PTGS2DHODHGAAMEN1KMT2A
SCHEMBL8666701 0.68 KDM4E (0.44) PTGS2DHODHCYP1A2GAAMEN1
SCHEMBL11564097 0.67 GABRA2 (0.46) DHODHCYP1A2PDE3BPDE3ANR1H2
SCHEMBL4416813 0.67 BRD4 (0.48) PTGS2DHODHCYP1A2PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811445-A ANGIOTENSIN II INHIBITORS ROUSSEL UCLAF (FR) 1998-09-22 US disclosed