SCHEMBL8666701

SCHEMBL8666701

Cc1nc(-c2ccc(-c3ccccc3)cc2)c(C(C(=O)O)C(F)(F)F)[nH]1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
HPGD P15428 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DHODH Q02127 6/20 0.40
CYP1A2 P05177 1/20 0.39
PDE2A O00408 1/20 0.38
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
ALDH1A1 P00352 2/20 0.36
GLA P06280 2/20 0.36
GAA P10253 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
ACMSD Q8TDX5 1/20 0.36
PTGS2 P35354 1/20 0.36
NTRK1 P04629 1/20 0.35
POLB P06746 1/20 0.35
PIN1 Q13526 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8666896 0.79 KDM4E (0.44) KDM4EHPGDSMN1; SMN2DHODHPDE2A
SCHEMBL4879884 0.71 KDM4E (0.59) KDM4EHPGDSMN1; SMN2DHODHCYP1A2
SCHEMBL8666901 0.68 PTGS2 (0.42) DHODHCYP1A2GAAKMT2AMEN1
SCHEMBL6547467 0.68 KDM4E (0.50) KDM4EHPGDSMN1; SMN2DHODHCYP1A2
SCHEMBL5762947 0.67 KDM4E (0.62) KDM4EHPGDSMN1; SMN2DHODHCYP1A2
SCHEMBL27653921 0.67 HPGD (0.58) KDM4EHPGDSMN1; SMN2DHODHCYP1A2
SCHEMBL8666893 0.67 PTGS2 (0.39) DHODHCYP1A2GAAKMT2AMEN1
SCHEMBL8666707 0.67 COMT (0.42) DHODHKMT2APTGS2
SCHEMBL7601774 0.64 HPGD (0.68) KDM4EHPGDSMN1; SMN2CYP1A2ALDH1A1
SCHEMBL5823944 0.64 KDM4E (0.53) KDM4EHPGDSMN1; SMN2CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811445-A ANGIOTENSIN II INHIBITORS ROUSSEL UCLAF (FR) 1998-09-22 US disclosed