SCHEMBL8667329

SCHEMBL8667329

O=C(O)CCC1CCc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.43
FFAR1 O14842 1/20 0.41
HSP90AA1 P07900 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HTR6 P50406 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
CYP1A2 P05177 1/20 0.40
PPARD Q03181 2/20 0.39
PNMT P11086 1/20 0.39
TBXA2R P21731 1/20 0.39
PPARA Q07869 1/20 0.38
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6668520 0.86 FFAR1 (0.55) GRIN2BFFAR1PPARDPPARA
SCHEMBL6839634 0.79 ESR1 (0.57) FFAR1MAPTHTR6PPARDPPARA
SCHEMBL8702101 0.77 GRIN2B (0.42) GRIN2BHSP90AA1PNMT
SCHEMBL9014699 0.75 PNMT (0.40) GRIN2BHSP90AA1HTR6PNMT
SCHEMBL1567103 0.74 MTNR1A (0.56) FFAR1HTR6L3MBTL1PPARD
SCHEMBL8667327 0.74 PNMT (0.50) HSP90AA1ALDH1A1MAPTPNMT
SCHEMBL8669494 0.73 MTNR1A (0.59) FFAR1CYP1A2
SCHEMBL2244560 0.71 LAP3 (0.48) GRIN2BHSP90AA1ALDH1A1MAPTPNMT
SCHEMBL8548146 0.71 PNMT (0.44) GRIN2BHSP90AA1ALDH1A1MAPTPNMT
SCHEMBL7214649 0.71 PNMT (0.48) GRIN2BHSP90AA1PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721234-A TREATING CONVULSIONS, ANXIETY, CEREBRAL HYPOXIA/ISCHEMIA, PARKINSON*S DISEASE WARNER-LAMBERT COMPANY (US) 1998-02-24 US disclosed
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO disclosed