SCHEMBL9014699

SCHEMBL9014699

O=[N+]([O-])c1ccc2c(c1)CCCC2CCBr

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PNMT P11086 3/20 0.40
NR3C1 P04150 1/20 0.40
HTR6 P50406 7/20 0.39
HSP90AA1 P07900 1/20 0.39
GRIN2B Q13224 2/20 0.38
CHRNA7 P36544 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
ADRA2A P08913 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014643 0.78 TERT (0.38) HSP90AA1SMN1; SMN2CHRNB4CHRNA3NOS3
SCHEMBL8667329 0.75 GRIN2B (0.43) PNMTHTR6HSP90AA1GRIN2B
SCHEMBL8702101 0.72 GRIN2B (0.42) PNMTHSP90AA1GRIN2BCHRNB2CHRNB4
SCHEMBL8548146 0.72 PNMT (0.44) PNMTHSP90AA1GRIN2BCHRNA7SMN1; SMN2
SCHEMBL10407545 0.72 HSP90AA1 (0.38) HSP90AA1SMN1; SMN2CHRNB4CHRNA3MEN1
SCHEMBL10551218 0.71 CYP19A1 (0.54)
SCHEMBL6668520 0.71 FFAR1 (0.55) GRIN2B
SCHEMBL9014412 0.70 KCNH2 (0.52)
SCHEMBL7509358 0.70 HSP90AA1 (0.47) PNMTHSP90AA1GRIN2BCHRNB2CHRNB4
SCHEMBL2244560 0.69 LAP3 (0.48) PNMTHSP90AA1GRIN2BCHRNA7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed