SCHEMBL8669271

SCHEMBL8669271

Cc1cc(Oc2cc(Cl)c(Cl)cc2Br)c(Cl)c(C)c1NC(=S)NC(=O)c1ccccc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.47
KDM4E B2RXH2 4/20 0.47
HPGD P15428 3/20 0.47
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
ALDH1A1 P00352 10/20 0.44
NPC1 O15118 4/20 0.44
KMT2A Q03164 6/20 0.41
MEN1 O00255 2/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
RAB9A P51151 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ALOX12 P18054 2/20 0.40
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657012 0.91 MAPT (0.45) MAPTKDM4EHPGDCRHBPCRHR2
SCHEMBL8660912 0.91 KMT2A (0.43) MAPTKDM4EHPGDALDH1A1NPC1
SCHEMBL8663047 0.87 CRHBP (0.47) MAPTKDM4EHPGDCRHBPCRHR2
SCHEMBL8657910 0.87 PNLIP (0.48) MAPTKDM4EHPGDCRHBPCRHR2
SCHEMBL8656183 0.84 POLB (0.39) MAPTCRHBPCRHR2ALDH1A1KMT2A
SCHEMBL8661113 0.84 KMT2A (0.43) MAPTKDM4EHPGDALDH1A1NPC1
SCHEMBL8665622 0.83 MAPT (0.51) MAPTKDM4EHPGDCRHBPCRHR2
SCHEMBL8658928 0.82 ALDH1A1 (0.49) MAPTHPGDALDH1A1NPC1KMT2A
SCHEMBL8658214 0.82 KMT2A (0.46) MAPTKDM4EHPGDALDH1A1NPC1
SCHEMBL8660959 0.82 PYGL (0.47) MAPTNPC1KMT2AMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed