SCHEMBL8672012

SCHEMBL8672012

C1=C(c2ccccc2)CCN(CCCCc2cc3ccccc3[nH]2)C1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.56
PARP1 P09874 4/20 0.55
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
HTR1A P08908 1/20 0.53
MAPT P10636 1/20 0.53
CYP2C9 P11712 1/20 0.53
DRD2 P14416 1/20 0.53
TSHR P16473 1/20 0.53
DRD4 P21917 1/20 0.53
CYP2C19 P33261 1/20 0.53
DRD3 P35462 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
HRH3 Q9Y5N1 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8683088 0.84 DRD4 (0.60) PARP1MAPTDRD2DRD4DRD3
SCHEMBL9775955 0.77 HRH3 (0.78) SIGMAR1HRH3
SCHEMBL3990045 0.76 HRH3 (0.63) SIGMAR1DRD2DRD3HRH3
SCHEMBL10969078 0.76 HTR1A (0.60) SIGMAR1PARP1CYP1A2CYP3A4HTR1A
SCHEMBL10967600 0.75 TDP1 (0.64) SIGMAR1PARP1CYP1A2CYP3A4HTR1A
SCHEMBL8871095 0.74 HTR1A (0.61) SIGMAR1CYP1A2CYP3A4HTR1AMAPT
SCHEMBL8688791 0.74 CHRNA7 (0.84) SIGMAR1PARP1CYP1A2CYP3A4TSHR
SCHEMBL9582455 0.73 PARP1 (0.56) SIGMAR1PARP1CYP1A2CYP3A4HTR1A
SCHEMBL8875223 0.73 PARP1 (0.58) PARP1CYP3A4MAPTDRD2TSHR
SCHEMBL7297566 0.73 SIGMAR1 (0.63) SIGMAR1PARP1HTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731331-A Tetrahydropyridine-(or 4-hydroxypiperidine) alkylazoles LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1998-03-24 US disclosed