SCHEMBL8672247

SCHEMBL8672247

Cc1c(O)cccc1C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)C[C@H](Cc1ccccc1)NC(=O)c1cccc(N)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.42
MME P08473 1/20 0.42
MMEL1 Q495T6 1/20 0.42
BACE1 P56817 7/20 0.40
CTRB1 P17538 1/20 0.40
BACE2 Q9Y5Z0 4/20 0.40
CTSD P07339 3/20 0.40
PIN1 Q13526 1/20 0.39
HPGDS O60760 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6927619 0.88 CTRB1 (0.50) CCR1MMEMMEL1BACE1CTRB1
SCHEMBL8670883 0.87 MAPK1 (0.44) CCR1BACE1NPC1RAB9A
SCHEMBL8669429 0.81 PSMB5 (0.44) CCR1BACE1BACE2CTSD
SCHEMBL8668860 0.80 ATM (0.49) BACE1
Hydrochloric Acid SCHEMBL8667609 0.80 PSMB5 (0.43) CCR1BACE1BACE2CTSD
SCHEMBL6929977 0.80 HPGDS (0.52) CCR1MMEMMEL1BACE1CTRB1
Hydrochloric Acid SCHEMBL8897869 0.78 CCR1 (0.43) CCR1BACE1BACE2CTSD
SCHEMBL8673190 0.76 CYP3A4 (0.54) CCR1CTRB1
SCHEMBL6924224 0.76 NPC1 (0.49) CCR1BACE1CTRB1BACE2CTSD
SCHEMBL5699585 0.75 PYGL (0.47) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763464-A TREATING HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-06-09 US disclosed
WO-1997019061-A1 RETROVIRAL AGENTS CONTAINING ANTHRANILAMIDE, SUBSTITUTED BENZAMIDE AND OTHER SUBUNITS, AND METHODS OF USING SAME THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1997-05-29 WO disclosed