SCHEMBL6929977

SCHEMBL6929977

O=C(N[C@@H](Cc1ccccc1)C[C@H](O)[C@H](Cc1ccccc1)NC(=O)c1cccc(O)c1)c1cccc(O)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 3/20 0.52
CCR1 P32246 4/20 0.51
CTRB1 P17538 1/20 0.50
MME P08473 1/20 0.48
MMEL1 Q495T6 1/20 0.48
BACE1 P56817 5/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GPR132 Q9UNW8 1/20 0.46
PIN1 Q13526 3/20 0.45
CTSD P07339 1/20 0.45
BACE2 Q9Y5Z0 1/20 0.45
CTSL P07711 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6927619 0.88 CTRB1 (0.50) HPGDSCCR1CTRB1MMEMMEL1
SCHEMBL6929416 0.85 HPGDS (0.58) HPGDSCCR1CTRB1BACE1KDM4E
SCHEMBL6931268 0.85 HPGDS (0.58) HPGDSCCR1CTRB1BACE1KDM4E
SCHEMBL6925409 0.85 HPGDS (0.58) HPGDSCCR1CTRB1BACE1KDM4E
SCHEMBL14005615 0.82 HPGDS (0.58) HPGDSCTRB1MMEMMEL1BACE1
SCHEMBL8672247 0.80 CCR1 (0.42) HPGDSCCR1CTRB1MMEMMEL1
SCHEMBL8670883 0.76 MAPK1 (0.44) CCR1BACE1ALDH1A1
SCHEMBL3497782 0.76 GPR132 (0.70) HPGDSGPR132
SCHEMBL28592116 0.76 GPR132 (0.70) HPGDSGPR132
SCHEMBL8773564 0.75 HPGDS (0.51) HPGDSCTRB1MMEMMEL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0801640-B1 2,5-DIAMINO-3,4-DISUBSTITUTED-1,6-DIPHENYLHEXANE ISOSTERES COMPRISING BENZAMIDE, SULFONAMIDE AND ANTHRANILAMIDE SUBUNITS AND METHODS OF USING SAME USA (US) 2003-03-26 EP claimed