SCHEMBL8680676

SCHEMBL8680676

COc1cccc(CCc2ccccc2)c1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.61
PTGS2 P35354 1/20 0.61
ABCB1 P08183 6/20 0.59
ABCG2 Q9UNQ0 2/20 0.57
IDO1 P14902 1/20 0.54
CALM1 P0DP23 1/20 0.54
HTR1A P08908 2/20 0.50
DRD2 P14416 2/20 0.50
LMNA P02545 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
ALOX12 P18054 1/20 0.50
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TAAR1 Q96RJ0 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9771763 0.84 CALM1 (0.69) ALOX5PTGS2IDO1CALM1HTR1A
SCHEMBL7709750 0.84 ALOX5 (0.55) ALOX5PTGS2ABCB1ABCG2IDO1
SCHEMBL7335269 0.83 ABCB1 (0.80) ABCB1ABCG2HTR1ADRD2TAAR1
SCHEMBL11711401 0.82 BCHE (0.66) LMNAKDM4ETAAR1
SCHEMBL30166692 0.82 BCHE (0.66) LMNAKDM4ETAAR1
SCHEMBL9423904 0.81 HTR1A (0.48) HTR1ADRD2ALDH1A1HPGDALOX15
SCHEMBL21030103 0.81 ABCB1 (0.77) ABCB1ABCG2HTR1ADRD2
SCHEMBL23748452 0.80 ALOX5 (0.77) ALOX5PTGS2IDO1CALM1LMNA
Benzyl Alcohol SCHEMBL27748093 0.79 ALOX5 (0.69) ALOX5PTGS2IDO1CALM1
SCHEMBL3252306 0.79 ABCB1 (0.59) ABCB1ABCG2HTR1ADRD2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110831584-B Targeted drug rescue with novel compositions, combinations and methods thereof 埃克塞瓦有限责任公司 2023-03-10 CN disclosed
EP-3618819-A1 TARGETED DRUG RESCUE WITH NOVEL COMPOSITIONS, COMBINATIONS, AND METHODS THEREOF Exciva GmbH (DE) 2020-03-11 EP disclosed
CN-110831584-A Targeted drug rescue with novel compositions, combinations and methods thereof 埃克塞瓦有限责任公司 2020-02-21 CN disclosed
WO-2018204713-A1 TARGETED DRUG RESCUE WITH NOVEL COMPOSITIONS, COMBINATIONS, AND METHODS THEREOF EXCIVA UG (HAFTUNGSBESCHRÄNKT) (DE) 2018-11-08 WO disclosed
US-5843983-A Diphenylethane compounds containing a saturated heterocyclic group, their preparation, and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1998-12-01 US disclosed
EP-0790235-A1 Diaryl alkane derivatives containing an alicyclic group, their preparation and their therapeutic and prophylactic uses SANKYO COMPANY LIMITED (JP) 1997-08-20 EP disclosed