SCHEMBL8686290

SCHEMBL8686290

COc1ccc(CNc2ncc(CC(=O)O)cn2)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
CA5A P35218 1/20 0.51
GAA P10253 6/20 0.50
TDP1 Q9NUW8 3/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ACHE P22303 3/20 0.49
APP P05067 2/20 0.49
POLB P06746 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
TPH1 P17752 1/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8686297 0.85 L3MBTL1 (0.55) ALDH1A1GAAMEN1KMT2AACHE
SCHEMBL8682662 0.83 ALDH1A1 (0.55) ALDH1A1GAATDP1MEN1KMT2A
SCHEMBL8686294 0.82 MAPK8 (0.54) ALDH1A1CA5AGAATDP1TSHR
SCHEMBL30049382 0.80 GAA (0.74) ALDH1A1CA5AGAATDP1TSHR
SCHEMBL153055 0.80 GAA (0.74) ALDH1A1CA5AGAATDP1TSHR
SCHEMBL27952523 0.78 GAA (0.72) ALDH1A1CA5AGAATDP1TSHR
Hydrochloric Acid SCHEMBL2530820 0.78 GAA (0.72) ALDH1A1CA5AGAATDP1TSHR
SCHEMBL21328339 0.75 CA5A (0.56) ALDH1A1CA5AGAATDP1TSHR
SCHEMBL21328347 0.74 CA5A (0.66) ALDH1A1CA5AGAATDP1TSHR
SCHEMBL21328344 0.74 GAA (0.70) ALDH1A1CA5AGAATDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719187-A Compounds having a guanidine structure and pharmaceutical composition containing same CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE(CNRS) (FR) 1998-02-17 US disclosed
US-5480884-A Compounds having a guanidine structure CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 1996-01-02 US disclosed
EP-0572635-A1 NOVEL COMPOUNDS HAVING A GUANIDINE STRUCTURE AND PHARMACEUTICAL COMPOSITION CONTAINING SAME. CENTRE NAT RECH SCIENT (FR) 1993-12-08 EP disclosed
EP-0572635-A4 NOVEL COMPOUNDS HAVING A GUANIDINE STRUCTURE AND PHARMACEUTICAL COMPOSITION CONTAINING SAME. CENTRE NAT RECH SCIENT (FR) 1993-09-17 EP disclosed
WO-1993010102-A1 NOVEL COMPOUNDS HAVING A GUANIDINE STRUCTURE AND PHARMACEUTICAL COMPOSITION CONTAINING SAME CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S) (FR) 1993-05-27 WO disclosed