SCHEMBL8690686

SCHEMBL8690686

CCOC(=O)CC[C@H](CCc1ccccc1)N(C(=O)[C@@H](N)Cc1ccccc1)C(=O)N1CCOCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
CTSL P07711 2/20 0.42
CTSB P07858 2/20 0.42
POLB P06746 2/20 0.40
FKBP1A P62942 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TMPRSS11D O60235 1/20 0.39
CTRL P40313 1/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 1/20 0.39
PSMB5 P28074 5/20 0.39
PSMB11 A5LHX3 1/20 0.38
PSMD11 O00231 1/20 0.38
PSMD12 O00232 1/20 0.38
PSMD14 O00487 1/20 0.38
PSMA7 O14818 1/20 0.38
PSMD3 O43242 1/20 0.38
CYP3A4 P08684 1/20 0.38
PSMC3 P17980 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8690672 0.79 PPID (0.42) ALDH1A1POLB
SCHEMBL8400709 0.75 FKBP1A (0.41) ALDH1A1CTSLCTSBPOLBFKBP1A
SCHEMBL4314424 0.69 CTSL (0.40) ALDH1A1CTSLCTSBTSHRCTSS
SCHEMBL9554848 0.69 FKBP1A (0.55) ALDH1A1CTSLCTSBPOLBFKBP1A
SCHEMBL9554857 0.69 FKBP1A (0.55) ALDH1A1CTSLCTSBPOLBFKBP1A
SCHEMBL7356293 0.67 FKBP1A (0.43) ALDH1A1CTSLCTSBPOLBFKBP1A
SCHEMBL7356298 0.67 FKBP1A (0.43) ALDH1A1CTSLCTSBPOLBFKBP1A
SCHEMBL21214616 0.67 ALOX5 (0.47) ALDH1A1POLBLMNAL3MBTL1
SCHEMBL6163356 0.67 HDAC8 (0.64) ALDH1A1FKBP1AMEN1KMT2ATSHR
SCHEMBL6052947 0.67 HDAC8 (0.64) ALDH1A1FKBP1AMEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776718-A Reversible protease inhibitors ARRIS PHARMACEUTICAL CORPORATION (US) 1998-07-07 US claimed
US-5776718-A Reversible protease inhibitors ARRIS PHARMACEUTICAL CORPORATION (US) 1998-07-07 US disclosed