SCHEMBL8690909

SCHEMBL8690909

O=C(c1ccccc1)c1cccnc1NCc1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
AURKA O14965 1/20 0.50
RPS6KB1 P23443 1/20 0.50
VNN1 O95497 4/20 0.49
DHODH Q02127 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
LMNA P02545 2/20 0.48
GAA P10253 1/20 0.48
HTT P42858 1/20 0.48
MAPK1 P28482 1/20 0.47
HIF1A Q16665 1/20 0.47
PDE5A O76074 2/20 0.47
NPC1 O15118 2/20 0.47
POLB P06746 2/20 0.47
RAB9A P51151 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554912 0.83 RPS6KB1 (0.65) MAOAMAOBAURKARPS6KB1HDAC3
SCHEMBL31204891 0.83 RPS6KB1 (0.65) MAOAMAOBAURKARPS6KB1HDAC3
SCHEMBL8696115 0.81 DHODH (0.52) DHODHLMNAGAAHTTNPC1
SCHEMBL8692447 0.79 KDM4E (0.68) DHODHLMNAGAAHTTNPC1
SCHEMBL8693733 0.77 DHODH (0.57) DHODHGAAHTTNPC1RAB9A
SCHEMBL1632005 0.77 CYP1A2 (0.54) SMN1; SMN2LMNAGAAHTTNPC1
SCHEMBL8694084 0.75 DHODH (0.76) DHODHSMN1; SMN2LMNAGAAHTT
SCHEMBL9842635 0.75 RAB9A (0.68) DHODHGAAHTTNPC1RAB9A
SCHEMBL29664470 0.74 MAOA (0.56) MAOAMAOBAURKARPS6KB1HDAC3
SCHEMBL18394876 0.74 MAOA (0.56) MAOAMAOBAURKARPS6KB1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1043993-C Nonel naphthyridine derivatives and medical composition thereof YAMANOUCHI PHARMA CO LTD (JP) 1999-07-07 CN disclosed
US-5817670-A RESPIRATORY SYSTEM DISORDERS, ORGAN TRANSPLANTATION, ANTITUMOR AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1998-10-06 US disclosed
CN-1156455-A Nonel naphthyridine derivatives and medical composition thereof YAMANOUCHI PHARMACUEITCAL CO L (JP) 1997-08-06 CN disclosed
EP-0779292-A1 NOVEL NAPHTHYRIDINE DERIVATIVE AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1997-06-18 EP disclosed