SCHEMBL8692197

SCHEMBL8692197

COc1ccc(-c2c(Cl)cnn2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.50
KDM4E B2RXH2 2/20 0.50
GAA P10253 2/20 0.50
ALDH1A1 P00352 5/20 0.49
NPSR1 Q6W5P4 3/20 0.49
LMNA P02545 2/20 0.49
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
NPBWR1 P48145 4/20 0.43
KMT2A Q03164 2/20 0.42
AURKA O14965 1/20 0.42
PRKAB2 O43741 1/20 0.42
PRKAG1 P54619 1/20 0.42
PRKAA2 P54646 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAG3 Q9UGI9 1/20 0.42
PRKAG2 Q9UGJ0 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688508 0.87 PTGS1 (0.49) HTTKDM4EGAAALDH1A1NPSR1
SCHEMBL8689251 0.86 ALDH1A1 (0.42) HTTKDM4EGAAALDH1A1NPSR1
SCHEMBL8639252 0.86 LMNA (0.48) HTTKDM4EGAAALDH1A1NPSR1
SCHEMBL8693823 0.86 PTGS2 (0.41) HTTKDM4EGAAALDH1A1KEAP1
SCHEMBL8689434 0.86 ALDH1A1 (0.49) HTTKDM4EGAAALDH1A1NPSR1
SCHEMBL8691901 0.85 PTGS2 (0.46) HTTKDM4EGAAALDH1A1LMNA
SCHEMBL8693263 0.84 NPSR1 (0.46) KDM4EGAAALDH1A1NPSR1LMNA
SCHEMBL8691135 0.83 HTT (0.47) HTTKDM4EGAAALDH1A1NPSR1
SCHEMBL8688904 0.82 ACLY (0.40) KDM4EGAAKMT2AMAPTMEN1
Benzenesulfonamide SCHEMBL8157094 0.81 PTGS2 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed