SCHEMBL8696594

SCHEMBL8696594

CNC(=O)Nc1cc(NC(=O)CCCc2ccccc2)ccc1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.55
RAB9A P51151 5/20 0.55
POLB P06746 1/20 0.55
TRPV1 Q8NER1 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
MAPT P10636 3/20 0.52
NFKB1 P19838 2/20 0.52
NFKB2 Q00653 2/20 0.52
RELA Q04206 2/20 0.52
ALDH1A1 P00352 2/20 0.52
ALOX15 P16050 1/20 0.52
MAPK1 P28482 1/20 0.52
MCL1 Q07820 1/20 0.52
LMNA P02545 1/20 0.51
HDAC1 Q13547 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8699518 0.79 ALDH1A1 (0.44) NPC1RAB9APOLBSMN1; SMN2MAPT
SCHEMBL8701009 0.76 ALOX5 (0.46) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL101223 0.76 HDAC1 (0.51) NPC1RAB9APOLBTRPV1SMN1; SMN2
SCHEMBL8701679 0.75 HDAC1 (0.57) NPC1RAB9ATRPV1SMN1; SMN2MAPT
SCHEMBL99412 0.74 HCAR2 (0.47) NPC1RAB9APOLBTRPV1SMN1; SMN2
SCHEMBL101227 0.73 NPC1 (0.45) NPC1RAB9APOLBTRPV1SMN1; SMN2
SCHEMBL99703 0.73 NPC1 (0.58) NPC1RAB9APOLBTRPV1SMN1; SMN2
SCHEMBL19501635 0.73 TRPV1 (0.77) NPC1RAB9APOLBTRPV1SMN1; SMN2
SCHEMBL101623 0.73 HDAC2 (0.48) TRPV1SMN1; SMN2MAPTALDH1A1HDAC1
SCHEMBL15822177 0.73 HDAC1 (0.47) NPC1RAB9APOLBTRPV1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726319-A Biphenyl substituted dipeptide analogs promote release of growth hormone MERCK & CO., INC. (US) 1998-03-10 US disclosed