SCHEMBL8697482

SCHEMBL8697482

N#Cc1ccc(C(O)c2cncnc2)c(F)c1-c1cc2ccccc2o1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.33
CYP2A6 P11509 1/20 0.33
PRKCQ Q04759 1/20 0.33
PRKCD Q05655 1/20 0.33
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
METAP2 P50579 1/20 0.32
MKNK1 Q9BUB5 3/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
ALOX5 P09917 1/20 0.30
ADK P55263 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8704175 0.89 CYP2A6 (0.34) CYP19A1CYP2A6PRKCQPRKCDCYP11B1
SCHEMBL8697485 0.81 CYP11B1 (0.34) CYP11B1CYP11B2KDM4EALDH1A1MAPT
SCHEMBL8696314 0.78 CYP19A1 (0.41) CYP19A1CYP2A6PRKCQPRKCDMETAP2
SCHEMBL8696579 0.74 MAOB (0.46) METAP2MKNK1MAOAMAOBALOX5
SCHEMBL8698524 0.69 FLT1 (0.33) CYP11B1CYP11B2KDM4EALDH1A1MAPT
SCHEMBL24621094 0.69 CYP19A1 (0.42) CYP19A1METAP2KDM4ETDP1NPC1
SCHEMBL8702186 0.67 CYP19A1 (0.47) CYP19A1CYP2A6KDM4EALDH1A1NPC1
SCHEMBL8698118 0.66 CYP11B1 (0.33) CYP11B1CYP11B2
SCHEMBL8700537 0.66 CYP19A1 (0.47) CYP19A1CYP2A6MAOAMAOBMAPT
SCHEMBL8700378 0.65 MAOB (0.46) CYP19A1METAP2MAOAMAOBALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO claimed