SCHEMBL8704175

SCHEMBL8704175

N#Cc1ccc(C(F)c2cncnc2)c(F)c1-c1cc2ccccc2o1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.34
CYP19A1 P11511 3/20 0.34
PRKCQ Q04759 1/20 0.33
PRKCD Q05655 1/20 0.33
CYP11B1 P15538 3/20 0.32
CYP11B2 P19099 3/20 0.32
METAP2 P50579 1/20 0.32
MKNK1 Q9BUB5 3/20 0.32
F2RL3 Q96RI0 3/20 0.32
ADK P55263 1/20 0.31
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697482 0.89 CYP19A1 (0.33) CYP2A6CYP19A1PRKCQPRKCDCYP11B1
SCHEMBL8697941 0.81 CYP11B1 (0.34) CYP11B1CYP11B2
SCHEMBL8700378 0.75 MAOB (0.46) CYP19A1METAP2F2RL3NPC1RAB9A
SCHEMBL8697485 0.69 CYP11B1 (0.34) CYP11B1CYP11B2MAPT
SCHEMBL8696314 0.68 CYP19A1 (0.41) CYP2A6CYP19A1PRKCQPRKCDMETAP2
SCHEMBL8702186 0.68 CYP19A1 (0.47) CYP2A6CYP19A1NPC1RAB9AMAPT
SCHEMBL8700537 0.67 CYP19A1 (0.47) CYP2A6CYP19A1MAPT
SCHEMBL8698606 0.65 ATM (0.32)
SCHEMBL1462351 0.64 MAOB (0.46) CYP2A6PRKCQPRKCDMETAP2NPC1
SCHEMBL19180722 0.64 MAOB (0.56) CYP19A1METAP2NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO disclosed