SCHEMBL8698701

SCHEMBL8698701

CCCn1cc(C(=O)OCC)c(NC(=S)N(C2CCCCC2)C2CCCCC2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 3/20 0.43
NPC1 O15118 2/20 0.43
MAPK1 P28482 1/20 0.40
KDR P35968 1/20 0.38
MTOR P42345 1/20 0.38
KMT2A Q03164 4/20 0.37
TDP1 Q9NUW8 3/20 0.37
LMNA P02545 4/20 0.36
NPSR1 Q6W5P4 3/20 0.36
MEN1 O00255 2/20 0.36
S1PR2 O95136 1/20 0.36
XBP1 P17861 1/20 0.36
NR2F2 P24468 1/20 0.36
RAB9A P51151 1/20 0.36
PPP1CA P62136 1/20 0.36
MAPT P10636 2/20 0.36
TSHR P16473 2/20 0.36
PRNP P04156 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8694014 0.94 ALDH1A1 (0.42) ALDH1A1KDM4ENPC1MAPK1KDR
SCHEMBL8696169 0.91 ALDH1A1 (0.48) ALDH1A1KDM4ENPC1MAPK1KMT2A
SCHEMBL8692971 0.86 ALDH1A1 (0.42) ALDH1A1KDM4ENPC1MAPK1KDR
SCHEMBL8693502 0.85 ALDH1A1 (0.46) ALDH1A1KDM4ENPC1MAPK1KMT2A
SCHEMBL8696060 0.83 TEAD2 (0.37) ALDH1A1KDM4EKMT2ATDP1LMNA
SCHEMBL8696385 0.83 MAPT (0.52) ALDH1A1KDM4ENPC1MAPK1KMT2A
SCHEMBL8693972 0.82 ALDH1A1 (0.42) ALDH1A1KDM4EKMT2ATDP1LMNA
SCHEMBL8696502 0.81 RAB9A (0.44) ALDH1A1KDM4ENPC1MAPK1KMT2A
SCHEMBL8696980 0.80 TEAD2 (0.37) ALDH1A1KDM4EKMT2ATDP1LMNA
SCHEMBL8696094 0.78 TEAD2 (0.38) ALDH1A1KDM4EKMT2ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed