SCHEMBL8699266

SCHEMBL8699266

CCc1c([N+](=O)[O-])ccc(OC(=O)O)c1[Si](C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 2/20 0.37
ALDH1A1 P00352 5/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
PDK1 Q15118 1/20 0.33
HTT P42858 1/20 0.33
CASP6 P55212 1/20 0.33
GSTP1 P09211 1/20 0.32
GSTM2 P28161 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28721667 0.80 GSTP1 (0.41) ALDH1A1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL47790 0.79 TSHR (0.42) FBP1ALDH1A1MEN1KMT2ALMNA
SCHEMBL47791 0.79 TSHR (0.42) FBP1ALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL28016724 0.77 GAA (0.38) FBP1ALDH1A1MEN1KMT2ALMNA
SCHEMBL7968000 0.77 FBP1 (0.36) FBP1ALDH1A1MEN1KMT2ALMNA
SCHEMBL618822 0.75 TXNRD1 (0.39) FBP1ALDH1A1MEN1KMT2ALMNA
SCHEMBL27311411 0.74 ALDH1A1 (0.41) FBP1ALDH1A1MEN1KMT2ALMNA
SCHEMBL27837566 0.73 SIRT6 (0.44) ALDH1A1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL7357833 0.71 ALDH1A1 (0.33) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL27364415 0.71 CTSV (0.46) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294732-A Conformationally constrained, fully synthetic macrocyclic compounds POLYPHOR AG 2016-02-03 CN disclosed
CN-102471349-A Conformationally constrained, fully synthetic macrocyclic compounds POLYPHOR AG 2012-05-23 CN disclosed
WO-1998023586-A1 AROMATIC AMINOALCOHOLS AS 5HT1A ANTAGONISTS AND AS SEROTONIN REABSORPTION INHIBITORS PIERRE FABRE MEDICAMENT (FR) 1998-06-04 WO disclosed