SCHEMBL8699309

SCHEMBL8699309

COc1nc(C)c(C(C)C)cc1N(C(=O)O)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.36
LPAR1 Q92633 4/20 0.35
MAPT P10636 3/20 0.34
LMNA P02545 2/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPK14 Q16539 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
ATM Q13315 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HSP90AA1 P07900 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7628968 0.84 MEN1 (0.46) TSHRKMT2AMEN1POLBMAPT
SCHEMBL7626374 0.81 MEN1 (0.40) TSHRKMT2AMEN1POLBMAPT
SCHEMBL8706000 0.74 TSHR (0.44) TSHRKMT2AMEN1POLBMAPT
SCHEMBL8699760 0.72 ALDH1A1 (0.39) TSHRKMT2AMEN1POLBMAPT
SCHEMBL8699460 0.72 TSHR (0.39) TSHRKMT2AMEN1POLBMAPT
SCHEMBL8699808 0.72 NPC1 (0.39) TSHRKMT2AMEN1POLBMAPT
SCHEMBL27466604 0.72 ATM (0.52) TSHRKMT2AMEN1LMNASMN1; SMN2
SCHEMBL8706005 0.71 MEN1 (0.40) TSHRKMT2AMEN1POLBMAPT
SCHEMBL8699467 0.70 TSHR (0.36) TSHRKMT2AMEN1POLBMAPT
SCHEMBL8699064 0.69 L3MBTL1 (0.39) TSHRKMT2AMEN1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780472-A ANTITUMOR AGENTS SAMJIN PHARMACEUTICAZL CO., LTD. (KR) 1998-07-14 US disclosed
EP-0749425-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARM. CO., LTD. (KR) 1996-12-27 EP disclosed
WO-1996021648-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1996-07-18 WO disclosed