SCHEMBL8701419

SCHEMBL8701419

N=C(N)NC(=O)c1cc(-n2cccc2)ccc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
POLB P06746 2/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48
HSD17B10 Q99714 1/20 0.48
AOC2 O75106 4/20 0.42
F2 P00734 4/20 0.36
F10 P00742 4/20 0.36
PLAU P00749 4/20 0.36
PLAT P00750 4/20 0.36
RAB9A P51151 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
NPC1 O15118 1/20 0.36
DNMT1 P26358 1/20 0.36
CASP6 P55212 1/20 0.36
MCL1 Q07820 1/20 0.36
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
PPIA P62937 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8705142 0.81 ALDH1A1 (0.48) ALDH1A1KDM4EPOLBHPGDMAPK1
SCHEMBL21884446 0.80 KAT6A (0.43) ALDH1A1KDM4EMAPK1MAPTGAA
SCHEMBL8703970 0.80 SIRT6 (0.41) ALDH1A1KDM4EPOLBHPGDMAPK1
Hydrochloric Acid SCHEMBL8705159 0.79 SIRT6 (0.40) ALDH1A1KDM4EPOLBHPGDMAPK1
SCHEMBL8701429 0.77 ALDH1A1 (0.45) ALDH1A1KDM4EPOLBHPGDMAPK1
SCHEMBL8704862 0.77 AOC2 (0.65) ALDH1A1POLBHPGDAOC2RAB9A
SCHEMBL8705516 0.77 AOC2 (0.68) ALDH1A1AOC2RAB9AL3MBTL1NPC1
Hydrochloric Acid SCHEMBL8707141 0.76 AOC2 (0.63) ALDH1A1POLBHPGDAOC2RAB9A
Hydrochloric Acid SCHEMBL8700020 0.75 AOC2 (0.66) ALDH1A1AOC2RAB9AL3MBTL1NPC1
SCHEMBL130491 0.75 KDM4E (0.74) ALDH1A1KDM4EPOLBHPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5824691-A CARDIOVASCULAR, CEREBROVASCULAR, RENAL DISEASES; SHOCK, ARTERIOSCLEROSIS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-10-20 US disclosed