SCHEMBL8701556

SCHEMBL8701556

NCc1ccc(-c2ccccc2[N+](=O)[O-])cc1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.65
TDP1 Q9NUW8 2/20 0.65
LOXL2 Q9Y4K0 1/20 0.52
TAAR1 Q96RJ0 1/20 0.47
GSK3A P49840 2/20 0.46
GSK3B P49841 2/20 0.46
AURKA O14965 1/20 0.46
S100A4 P26447 2/20 0.45
PTPRC P08575 1/20 0.45
TSHR P16473 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
MGAM O43451 1/20 0.43
GAA P10253 1/20 0.43
SI P14410 1/20 0.43
MGAM2 Q2M2H8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SLC9A1 P19634 1/20 0.43
ADAMTS4 O75173 1/20 0.42
PTPN1 P18031 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785924 0.84 ALDH1A1 (0.67) ALDH1A1TDP1GSK3AGSK3BAURKA
SCHEMBL7833436 0.84 ALDH1A1 (0.57) ALDH1A1TDP1GSK3AGSK3BAURKA
SCHEMBL3956866 0.83 ALDH1A1 (0.65) ALDH1A1TDP1GSK3AGSK3BAURKA
SCHEMBL17468329 0.83 ALDH1A1 (0.65) ALDH1A1TDP1GSK3AGSK3BAURKA
SCHEMBL32679855 0.83 ALDH1A1 (0.70) ALDH1A1TDP1GSK3AGSK3BAURKA
SCHEMBL10712973 0.80 ALDH1A1 (0.71) ALDH1A1TDP1S100A4PTPRCTSHR
SCHEMBL98895 0.80 ALDH1A1 (0.56) ALDH1A1TDP1LOXL2TAAR1TSHR
SCHEMBL2958562 0.80 ALDH1A1 (0.92) ALDH1A1TDP1S100A4PTPRCTSHR
Benzylamine SCHEMBL27935314 0.80 LOXL2 (0.58) ALDH1A1TDP1LOXL2TSHRGAA
SCHEMBL30196067 0.79 ALDH1A1 (1.00) ALDH1A1TDP1S100A4PTPRCTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726319-A Biphenyl substituted dipeptide analogs promote release of growth hormone MERCK & CO., INC. (US) 1998-03-10 US disclosed
EP-0669830-A4 SUBSTITUTED DIPEPTIDE ANALOGS PROMOTE RELEASE OF GROWTH HORMONE. MERCK & CO INC (US) 1997-02-26 EP disclosed
EP-0669830-A1 SUBSTITUTED DIPEPTIDE ANALOGS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO. INC. (US) 1995-09-06 EP disclosed
US-5330989-A Heterocycles substituted with biphenyl-3-cyclobutene-1,2-dione derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1994-07-19 US disclosed
WO-1994011012-A1 SUBSTITUTED DIPEPTIDE ANALOGS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1994-05-26 WO disclosed