SCHEMBL8709162

SCHEMBL8709162

COc1cc(CC(C(=O)NS(=O)(=O)c2ccccc2)c2ccc3nsnc3c2)cc(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.45
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
ITGB3 P05106 1/20 0.39
ITGAV P06756 1/20 0.39
PPARA Q07869 1/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 2/20 0.38
GAA P10253 2/20 0.38
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
TACR1 P25103 1/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709051 0.92 MAPT (0.39) MAPTEGFRERBB2ITGB3ITGAV
SCHEMBL8705645 0.90 MEN1 (0.41) MAPTPPARANPC1RAB9ASMN1; SMN2
SCHEMBL8706237 0.89 ITGB3 (0.40) MAPTITGB3ITGAVNPC1RAB9A
SCHEMBL8709447 0.88 ITGB3 (0.48) MAPTEGFRERBB2ITGB3ITGAV
SCHEMBL8709683 0.87 ITGB3 (0.43) MAPTEGFRERBB2ITGB3ITGAV
SCHEMBL8709876 0.86 BCL2 (0.42) MAPTEGFRERBB2ITGB3ITGAV
SCHEMBL8706016 0.85 NPC1 (0.44) MAPTITGB3ITGAVNPC1RAB9A
SCHEMBL8712032 0.84 SLC7A5 (0.43) MAPTITGB3ITGAVSMN1; SMN2MEN1
SCHEMBL8709691 0.84 ITGB3 (0.39) MAPTEGFRERBB2ITGB3ITGAV
SCHEMBL8712259 0.84 BMP1 (0.43) MAPTEGFRERBB2PPARANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041515-A1 ENDOTHOLIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed