SCHEMBL8709691

SCHEMBL8709691

COC(=O)CC(C)c1ccc(CC(C(=O)NS(=O)(=O)c2ccccc2)c2ccc3nsnc3c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.39
ITGAV P06756 1/20 0.39
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
LARS1 Q9P2J5 1/20 0.37
PPARA Q07869 1/20 0.37
BCL2 P10415 1/20 0.36
TARS1 P26639 1/20 0.36
HDAC1 Q13547 1/20 0.36
MAPT P10636 3/20 0.36
REN P00797 1/20 0.36
SCN3A Q9NY46 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
POLB P06746 2/20 0.35
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PRSS1 P07477 1/20 0.35
GAA P10253 2/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709961 0.93 ITGB3 (0.36) ITGB3ITGAVEGFRERBB2PPARA
SCHEMBL8709789 0.91 MEN1 (0.39) ITGB3ITGAVPPARAMAPTMEN1
SCHEMBL8709447 0.88 ITGB3 (0.48) ITGB3ITGAVEGFRERBB2LARS1
SCHEMBL8709876 0.87 BCL2 (0.42) ITGB3ITGAVEGFRERBB2BCL2
SCHEMBL8709683 0.87 ITGB3 (0.43) ITGB3ITGAVEGFRERBB2LARS1
SCHEMBL8706743 0.85 TARS1 (0.39) ITGB3ITGAVEGFRERBB2LARS1
SCHEMBL8709162 0.84 MAPT (0.45) ITGB3ITGAVEGFRERBB2LARS1
SCHEMBL8712259 0.84 BMP1 (0.43) EGFRERBB2PPARAMAPTMEN1
SCHEMBL8706237 0.83 ITGB3 (0.40) ITGB3ITGAVMAPTPOLBHSD17B10
SCHEMBL8712032 0.82 SLC7A5 (0.43) ITGB3ITGAVMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041515-A1 ENDOTHOLIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed