SCHEMBL8709756

SCHEMBL8709756

FC(F)(F)Oc1cccc(-c2nsc(Cl)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.46
MPI P34949 1/20 0.46
S1PR1 P21453 1/20 0.45
XDH P47989 1/20 0.43
DYRK1A Q13627 2/20 0.42
KCNH2 Q12809 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.42
NPY5R Q15761 1/20 0.41
ADORA1 P30542 2/20 0.40
ADORA2A P29274 1/20 0.40
BACE1 P56817 1/20 0.40
DHODH Q02127 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
PIM1 P11309 2/20 0.39
ATR Q13535 1/20 0.39
PRMT1 Q99873 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14488342 0.82 CASP3 (0.51)
SCHEMBL14488273 0.81 CYP19A1 (0.56) DYRK1AADORA1ADORA2A
SCHEMBL9028816 0.78 CASP3 (0.52) S1PR1DYRK1AADORA2AHDAC1HDAC6
SCHEMBL3769512 0.75 KDM4E (0.42) GRM5ADORA1ADORA2A
SCHEMBL14488183 0.75 CYP19A1 (0.46) GRM5MPI
SCHEMBL8103598 0.73 DYRK1A (0.61) GRM5S1PR1XDHDYRK1AKCNH2
SCHEMBL8549187 0.72 HSD17B1 (0.68)
SCHEMBL14755837 0.72 ALDH1A1 (0.51)
SCHEMBL5244655 0.71 SMN1; SMN2 (0.47) DHODH
SCHEMBL16481833 0.71 L3MBTL1 (0.64) GRM5S1PR1XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998023155-A1 ARTHROPODICIDAL AND FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-06-04 WO disclosed
WO-1997000612-A1 ARTHROPODICIDAL AND FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1997-01-09 WO disclosed