SCHEMBL8710208

SCHEMBL8710208

CCOC(=O)CC1(c2ccccc2)C(=O)NCc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.48
MEN1 O00255 2/20 0.44
CYP1A2 P05177 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
APEX1 P27695 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GAA P10253 2/20 0.41
ALDH1A1 P00352 3/20 0.41
OPRM1 P35372 4/20 0.39
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
SLC22A1 O15245 1/20 0.38
SLC6A4 P31645 1/20 0.38
ADRA1A P35348 1/20 0.38
KCNH2 Q12809 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102535 0.72 ALDH1A1 (0.68) BRD4MEN1CYP1A2KMT2AGAA
SCHEMBL4851721 0.72 SIGMAR1 (0.42) BRD4KMT2ATSHRGAAALDH1A1
SCHEMBL8711235 0.68 KMT2A (0.37) MEN1CYP1A2KMT2APOLBTSHR
SCHEMBL2637139 0.68 GAA (0.53) BRD4MEN1KMT2AGAAALDH1A1
SCHEMBL9337866 0.67 GAA (0.59) BRD4MEN1KMT2AGAAALDH1A1
SCHEMBL7607750 0.66 SMN1; SMN2 (0.48) BRD4TSHRGAAALDH1A1LMNA
SCHEMBL735234 0.66 IDO1 (0.59) TSHRGAAALDH1A1LMNAMAPT
SCHEMBL26692976 0.66 MEN1 (0.46) MEN1KMT2AGAAALDH1A1OPRM1
SCHEMBL9666272 0.66 BRD4 (0.38) BRD4TSHRGAAALDH1A1OPRM1
SCHEMBL8368989 0.65 OPRM1 (0.62) GAAOPRM1OPRD1OPRK1SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998002432-A1 BICYCLIC COMPOUNDS FOR CONTROLLING MICTURITION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-22 WO disclosed