SCHEMBL8711235

SCHEMBL8711235

CCC(C(=O)O)C1(c2ccccc2)C(=O)NCc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37
APEX1 P27695 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
OPRM1 P35372 2/20 0.35
OPRK1 P41145 2/20 0.35
OPRL1 P41146 2/20 0.35
KIF11 P52732 4/20 0.35
EDNRA P25101 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA1A P35348 1/20 0.33
TP53 P04637 1/20 0.33
EDNRB P24530 1/20 0.32
MYC P01106 1/20 0.32
LMNA P02545 1/20 0.32
ADAMTS5 Q9UNA0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703449 0.72 LMNA (0.37) KMT2AMEN1KIF11HTR1AADRA1A
SCHEMBL8710208 0.68 BRD4 (0.48) KMT2AMEN1CYP1A2POLBTSHR
SCHEMBL8704259 0.68 KDM5A (0.42) KMT2AMEN1KIF11
SCHEMBL2512448 0.65 TSHR (0.42) POLBTSHROPRM1OPRL1LMNA
SCHEMBL21219221 0.63 THRB (0.44) KMT2AMEN1CYP1A2POLBAPEX1
SCHEMBL29506875 0.63 THRB (0.44) KMT2AMEN1CYP1A2POLBAPEX1
SCHEMBL6070188 0.62 ALDH1A1 (0.61) KMT2AMEN1TSHROPRM1KIF11
SCHEMBL23553895 0.62 CA12 (0.42) TSHRTDP1OPRM1OPRK1OPRL1
SCHEMBL30024606 0.62 CA12 (0.42) TSHRTDP1OPRM1OPRK1OPRL1
SCHEMBL30807380 0.62 OPRM1 (0.56) TSHRTDP1OPRM1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998002432-A1 BICYCLIC COMPOUNDS FOR CONTROLLING MICTURITION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-22 WO disclosed