SCHEMBL8710246

SCHEMBL8710246

COCOc1cc(C#N)c(Br)cc1C(=O)c1ncccc1OCOC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.40
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
GRM4 Q14833 1/20 0.35
APAF1 O14727 1/20 0.35
TDP2 O95551 1/20 0.35
NSD2 O96028 1/20 0.35
CASP3 P42574 1/20 0.35
PPP1CA P62136 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
SAE1 Q9UBE0 1/20 0.35
UBA2 Q9UBT2 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709829 0.87 XDH (0.40) XDHEGFRERBB2GRM4RAB9A
SCHEMBL8020333 0.85 XDH (0.45) XDHEGFRERBB2GRM4APAF1
SCHEMBL8709273 0.85 XDH (0.40) XDHGRM4ALDH1A1KDM4ERAB9A
SCHEMBL8709579 0.83 KDM4E (0.38) APAF1TDP2NSD2CASP3PPP1CA
SCHEMBL8715277 0.83 CLCN2 (0.38) GRM4APAF1TDP2NSD2CASP3
SCHEMBL8709782 0.83 SLC22A12 (0.40) XDHGRM4RAB9ANPC1LMNA
SCHEMBL8709054 0.79 CYP3A4 (0.47) ALDH1A1KDM4EMAPTCYP3A4
SCHEMBL8709890 0.78 RAB9A (0.37) ALDH1A1KDM4ERAB9ANPC1CHEK1
SCHEMBL8714963 0.76 PPIA (0.43) ALDH1A1NPC1LMNA
SCHEMBL8710268 0.76 XDH (0.43) XDHRAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed