SCHEMBL8020333

SCHEMBL8020333

COCOc1cccnc1C(=O)c1ccc(C#N)c(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.45
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HPGD P15428 2/20 0.36
EGFR P00533 2/20 0.36
CYP1A2 P05177 2/20 0.36
ERBB2 P04626 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
APAF1 O14727 1/20 0.34
NSD2 O96028 1/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710246 0.85 XDH (0.40) XDHALDH1A1NPC1RAB9AEGFR
SCHEMBL8024858 0.83 ALDH1A1 (0.39) ALDH1A1NPC1HPGDEGFRCYP1A2
SCHEMBL8020675 0.79 TDP1 (0.42) ALDH1A1NPC1RAB9AHPGDCYP1A2
SCHEMBL8709829 0.76 XDH (0.40) XDHNPC1RAB9AEGFRCYP1A2
SCHEMBL8709273 0.76 XDH (0.40) XDHALDH1A1NPC1RAB9AS1PR1
SCHEMBL8709782 0.72 SLC22A12 (0.40) XDHNPC1RAB9AHPGDS1PR1
SCHEMBL8709054 0.72 CYP3A4 (0.47) ALDH1A1CYP2D6CYP2C19CYP3A4
SCHEMBL8715277 0.72 CLCN2 (0.38) ALDH1A1RAB9AAPAF1NSD2CASP3
SCHEMBL8709579 0.72 KDM4E (0.38) ALDH1A1RAB9ACYP2D6CYP2C19APAF1
SCHEMBL8710268 0.70 XDH (0.43) XDHNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802187-B1 Hydroxypyridine derivatives, their production and their pharmaceutical use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-02-16 EP disclosed
US-5891895-A POTASSIUM CHANNEL MODULATORS; ANGINA PECTORIS; HYPERTENSIVEAGENTS; CARDIOVASCULAR, RESPIRATORY SYSTEM, BRAIN, GASTROINTESTINAL AND UROGENITAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0802187-A1 Hydroxypyridine derivatives, their production and their pharmaceutical use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-22 EP disclosed