SCHEMBL8711040

SCHEMBL8711040

COc1ccc(N2CCN(C)CC2)c(NC(=O)OC(C)(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 2/20 0.54
ALDH1A1 P00352 4/20 0.53
KDM4E B2RXH2 1/20 0.53
TSHR P16473 1/20 0.53
HTT P42858 1/20 0.51
KMT2A Q03164 6/20 0.50
MEN1 O00255 3/20 0.50
GAA P10253 3/20 0.49
F10 P00742 2/20 0.47
CSF1R P07333 1/20 0.46
BACE1 P56817 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716846 0.86 WDR5 (0.48) WDR5ALDH1A1KDM4ETSHRHTT
SCHEMBL8716619 0.84 WDR5 (0.51) WDR5ALDH1A1KDM4ETSHRHTT
SCHEMBL8908801 0.81 MAPK1 (0.57) ALDH1A1KDM4ETSHRHTTKMT2A
SCHEMBL13832429 0.79 BRPF1 (0.45) WDR5ALDH1A1KDM4EKMT2AMEN1
SCHEMBL8716632 0.79 KMT2A (0.46) WDR5ALDH1A1KMT2AMEN1GAA
SCHEMBL17857107 0.77 IRAK4 (0.51) TSHRKMT2APOLB
SCHEMBL19221922 0.76 ABL1 (0.46) WDR5ALDH1A1KDM4EKMT2AMEN1
SCHEMBL29823053 0.76 ABL1 (0.46) WDR5ALDH1A1KDM4EKMT2AMEN1
SCHEMBL4568017 0.76 GAA (0.50) HTTKMT2AMEN1GAAF10
SCHEMBL29991362 0.76 GAA (0.60) ALDH1A1KDM4ETSHRHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998031669-A1 NOVEL ARYLPIPERAZINE DERIVED FROM PIPERIDINE AS ANTIDEPRESSANT MEDICINES PIERRE FABRE MEDICAMENT (FR) 1998-07-23 WO disclosed