SCHEMBL8712010

SCHEMBL8712010

OC1C2CCN(CC2)C1C#Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP1B1 Q16678 1/20 0.38
GRM5 P41594 2/20 0.36
HRH3 Q9Y5N1 1/20 0.36
SLC18A3 Q16572 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8707234 0.87 HRH3 (0.37) GRM5HRH3KDM4E
SCHEMBL8920052 0.76 KMT2A (0.53) CYP1A2SLC18A3KDM4EMEN1NPC1
SCHEMBL8574139 0.75 CHRNA7 (0.50) CYP1A2GRM5
SCHEMBL8921220 0.75 MCHR1 (0.30)
Hydrochloric Acid SCHEMBL8578709 0.74 CHRNA7 (0.49) CYP1A2GRM5
SCHEMBL8921686 0.73 MEN1 (0.38) CYP1A2SLC18A3KDM4EMEN1NPC1
SCHEMBL8421878 0.72 CHRNA7 (0.36) SLC18A3
SCHEMBL8573706 0.70 TTR (0.41) CYP1A2GRM5HRH3KDM4ENPC1
SCHEMBL3259554 0.69 ALPL (0.34) HRH3SLC18A3KMT2A
SCHEMBL8520797 0.69 FFAR1 (0.38) SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770608-A ANTICHOLESTEROL AGENTS FOR TREATING CARDIOVASCULAR DISORDERS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1998-06-23 US disclosed