SCHEMBL8712930

SCHEMBL8712930

COCOc1cc(Cl)c(Br)cc1C(C#N)c1ncccc1OCOC

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
S1PR4 O95977 1/20 0.32
MAPT P10636 2/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KDM4E B2RXH2 1/20 0.30
EGFR P00533 1/20 0.30
ERBB2 P04626 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712772 0.84 EGFR (0.36) ALDH1A1MAPTHTTSMN1; SMN2KDM4E
SCHEMBL8715493 0.80 SGMS2 (0.37) ALDH1A1GAALMNAHPGDKDM4E
SCHEMBL8710153 0.74 EGFR (0.33) S1PR4EGFRERBB2
SCHEMBL8709739 0.69 CYP3A4 (0.32) EGFRERBB2
SCHEMBL8715277 0.68 CLCN2 (0.38) ALDH1A1POLBS1PR4MAPTLMNA
SCHEMBL31082087 0.67 MEN1 (0.35) ALDH1A1POLBGAANPSR1S1PR4
SCHEMBL17625811 0.67 LMNA (0.40) ALDH1A1POLBNPSR1MAPTLMNA
SCHEMBL8709673 0.66 CSNK2A1 (0.43)
SCHEMBL8715028 0.65 L3MBTL1 (0.38) ALDH1A1GAAS1PR4MAPTLMNA
SCHEMBL31082195 0.65 PLAU (0.35) ALDH1A1POLBNPSR1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed