SCHEMBL8713015

SCHEMBL8713015

Cc1nc2cccc3n(C[C@H]4CC[C@H](CNC(=O)C(F)(F)C(F)(F)F)CC4)c(=O)c1n23

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.34
HTR1A P08908 2/20 0.34
DRD2 P14416 2/20 0.34
DRD4 P21917 2/20 0.34
MDM2 Q00987 4/20 0.34
TP53 P04637 1/20 0.34
CKS1B P61024 4/20 0.33
SKP1 P63208 4/20 0.33
SKP2 Q13309 4/20 0.33
KCNH2 Q12809 2/20 0.33
GRM2 Q14416 1/20 0.32
RIPK1 Q13546 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
PTGER4 P35408 1/20 0.32
AVPR1B P47901 2/20 0.31
PDE5A O76074 1/20 0.31
PDE4A P27815 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713210 0.93 CKS1B (0.38) CNR2HTR1ADRD2DRD4MDM2
SCHEMBL7863439 0.79 DRD2 (0.34) CNR2HTR1ADRD2DRD4TP53
SCHEMBL7872441 0.79 DRD2 (0.33) CNR2HTR1ADRD2DRD4TP53
Hydrochloric Acid SCHEMBL8718961 0.77 ADORA3 (0.37) KCNH2GRM2ADORA3ADORA2APDE5A
SCHEMBL7871653 0.76 PDE5A (0.37) CNR2TP53KCNH2GRM2ADORA3
SCHEMBL7872489 0.76 DRD2 (0.38) CNR2DRD2ADORA3ADORA2APDE5A
Hydrochloric Acid SCHEMBL7872363 0.76 PDE5A (0.36) CNR2TP53KCNH2GRM2ADORA3
SCHEMBL8713886 0.75 HTR1A (0.34) HTR1ADRD2DRD4KCNH2
SCHEMBL8713955 0.75 ALDH1A1 (0.45) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7868708 0.75 GPR119 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826686-A2 Tricyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-04 EP disclosed