SCHEMBL8713416

SCHEMBL8713416

COc1ccc(N2C(=O)c3cnccc3C2C)cc1OCC1CCCC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
PDE4B Q07343 11/20 0.40
PDE4D Q08499 2/20 0.39
LMNA P02545 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
PDE4A P27815 1/20 0.38
PDE4C Q08493 1/20 0.38
CYP17A1 P05093 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712205 0.92 HTR2C (0.42) HTR2CHTR2BPDE4BPDE4DLMNA
SCHEMBL8714432 0.86 HTR2C (0.49) HTR2CHTR2BPDE4BPDE4DPDE4A
SCHEMBL8713534 0.85 LMNA (0.48) HTR2CHTR2BLMNACYP17A1
SCHEMBL8707491 0.82 HTR2C (0.49) HTR2CHTR2BPDE4BPDE4DPDE4A
SCHEMBL7695166 0.78 PDE4D (0.45) PDE4BPDE4DLMNAPDE4APDE4C
SCHEMBL8711411 0.77 PDE4D (0.44) PDE4BPDE4DLMNAPDE4APDE4C
SCHEMBL8712925 0.76 PDE4B (0.44) HTR2CHTR2BPDE4BPDE4DPDE4A
SCHEMBL8712036 0.75 RAB9A (0.54) HTR2CPDE4BPDE4DPDE4APDE4C
SCHEMBL8713070 0.74 PDE4B (0.43) HTR2CHTR2BPDE4BPDE4DPDE4A
SCHEMBL7696958 0.71 PDE4B (0.49) HTR2CHTR2BPDE4BPDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998042666-A1 NOVEL 3,4-DIALKOXYPHENYL DERIVATIVES AND THE USE THEREOF DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 1998-10-01 WO disclosed