SCHEMBL8713545

SCHEMBL8713545

O=C(Nc1cnc(Sc2cccc(-c3nnn[nH]3)c2)s1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.47
KDR P35968 2/20 0.41
SCD O00767 1/20 0.38
KMT2A Q03164 2/20 0.36
F2 P00734 3/20 0.35
F12 P00748 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
COMT P21964 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
MAPT P10636 3/20 0.35
PTPN5 P54829 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PRKD3 O94806 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044797 0.80 HDAC6 (0.41) HDAC6KDRSCDNPC1RAB9A
SCHEMBL8709996 0.80 HDAC6 (0.37) HDAC6KDRSCDNPC1RAB9A
SCHEMBL8714250 0.74 MAPK9 (0.44) KMT2ANPC1RAB9AMAPTNPSR1
SCHEMBL8045484 0.73 HDAC6 (0.57) HDAC6KDRSCDKMT2ANPC1
SCHEMBL8033612 0.71 HDAC6 (0.43) HDAC6KDRSCDNPC1RAB9A
SCHEMBL31680549 0.70 MMP2 (0.54) HDAC6KMT2ANPC1RAB9AMMP2
SCHEMBL8032616 0.69 SMN1; SMN2 (0.54) HDAC6KDRKMT2ANPC1RAB9A
SCHEMBL8032385 0.69 ALDH1A1 (0.48) HDAC6KDRKMT2ANPC1RAB9A
SCHEMBL2664555 0.69 HCAR3 (0.55) KMT2ANPC1RAB9AMAPTSMN1; SMN2
SCHEMBL8051066 0.68 RAB9A (0.44) HDAC6NPC1RAB9AMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed