SCHEMBL8713624

SCHEMBL8713624

O=[C]N(c1ccccc1)N1CCNCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.41
ADRB1 P08588 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR2A P28223 4/20 0.36
HTR2C P28335 3/20 0.36
HTR6 P50406 2/20 0.36
POLB P06746 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HTR1A P08908 2/20 0.35
HTR7 P34969 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718452 0.83 ADRB1 (0.44) SIGMAR1ADRB1HTR3AALDH1A1MEN1
SCHEMBL27418984 0.81 ALDH1A1 (0.40) ALDH1A1MEN1KMT2APOLBTSHR
SCHEMBL5774546 0.79 KMT2A (0.43) ALDH1A1MEN1KMT2APOLBTSHR
SCHEMBL8715074 0.76 PLD1 (0.45) ALDH1A1MEN1KMT2AHTR6USP2
SCHEMBL8719888 0.73 MAPT (0.31) SIGMAR1ADRB1HTR3EHTR3BHTR3A
SCHEMBL8716758 0.73 ADRB1 (0.32) SIGMAR1ADRB1HTR3EHTR3BHTR3A
SCHEMBL736136 0.72 SIGMAR1 (0.46) SIGMAR1ADRB1HTR3EHTR3BHTR3A
SCHEMBL21906494 0.72 SIGMAR1 (0.45) SIGMAR1ADRB1HTR3EHTR3BHTR3A
SCHEMBL27620685 0.72 SIGMAR1 (0.45) SIGMAR1ADRB1HTR3EHTR3BHTR3A
SCHEMBL28228488 0.72 SIGMAR1 (0.45) SIGMAR1ADRB1HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0822939-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 1998-02-11 EP disclosed
WO-1996034012-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed