SCHEMBL8715074

SCHEMBL8715074

O=[C]N(c1ccccn1)N1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 1/20 0.45
HTR7 P34969 2/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HTR1A P08908 1/20 0.37
TSHR P16473 2/20 0.36
HSD17B10 Q99714 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
SLC6A4 P31645 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713624 0.76 SIGMAR1 (0.41) HTR7ALDH1A1HTR1ATSHRHSD17B10
SCHEMBL31511748 0.74 PLD1 (0.43) PLD1HTR7ALDH1A1KDM4EHTR1A
SCHEMBL17329309 0.71 ALDH1A1 (0.43) PLD1ALDH1A1KDM4ETSHRHPGD
SCHEMBL4177502 0.71 PLD1 (0.43) PLD1HTR7ALDH1A1SMN1; SMN2
SCHEMBL8716758 0.68 ADRB1 (0.32) ALDH1A1CYP3A4CYP2D6HPGD
SCHEMBL8719888 0.68 MAPT (0.31)
SCHEMBL5113337 0.67 CYP2D6 (0.42) ALDH1A1KDM4ETSHRHSD17B10MEN1
SCHEMBL8718452 0.67 ADRB1 (0.44) HTR7ALDH1A1KDM4EHTR1ATSHR
SCHEMBL5773950 0.67 CYP2D6 (0.35) ALDH1A1KDM4EMEN1CYP3A4CYP2D6
SCHEMBL4557820 0.66 SIGMAR1 (0.41) PLD1HTR7ALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0822939-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 1998-02-11 EP disclosed
WO-1996034012-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed