SCHEMBL8715997

SCHEMBL8715997

O=Cc1ccc2oc3ccc(C=O)cc3c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.50
ALDH1A1 P00352 8/20 0.43
TSHR P16473 1/20 0.43
KDM4E B2RXH2 6/20 0.43
RAB9A P51151 4/20 0.43
PTGS2 P35354 1/20 0.43
KIF11 P52732 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
HSD17B10 Q99714 1/20 0.42
NPC1 O15118 4/20 0.40
POLB P06746 4/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
MAPT P10636 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
GFER P55789 1/20 0.39
HPGD P15428 3/20 0.38
ESR1 P03372 1/20 0.38
APEX1 P27695 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1420897 0.90 MAPT (0.53) CYP2A6ALDH1A1KDM4ERAB9AKIF11
SCHEMBL4966619 0.82 PARP10 (0.46) CYP2A6ALDH1A1TSHRKDM4ERAB9A
SCHEMBL1784133 0.81 MAOA (0.62) ALDH1A1KDM4ERAB9AKIF11HSD17B10
SCHEMBL9754623 0.81 CYP2A6 (0.65) CYP2A6ALDH1A1KDM4ETDP1HSD17B10
SCHEMBL6856438 0.81 CYP2A6 (0.45) CYP2A6ALDH1A1TSHRKDM4ERAB9A
SCHEMBL11337638 0.80 CDK9 (0.46) CYP2A6ALDH1A1TSHRKDM4ERAB9A
SCHEMBL29826652 0.80 KDM4E (0.44) CYP2A6ALDH1A1KDM4ERAB9APTGS2
SCHEMBL28086844 0.80 ALDH1A1 (0.48) CYP2A6ALDH1A1KDM4ERAB9APTGS2
SCHEMBL28950337 0.80 KDM4E (0.44) CYP2A6ALDH1A1KDM4ERAB9APTGS2
SCHEMBL13242794 0.80 ALDH1A1 (0.38) CYP2A6ALDH1A1KDM4ERAB9AKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP disclosed
US-5807974-A POLYARYLENEVINYLENE RESIN KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 1998-09-15 US disclosed
EP-0041675-B1 4-HALOGEN-5-(TRICHLOROMETHYL-PHENYL)-OXAZOLE DERIVATIVES, PROCESS FOR PREPARING THEM AND RADIATION-SENSITIVE COMPOSITIONS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-11 EP disclosed
US-4371607-A 4-Halogeno-5-(halogenomethyl-phenyl)-oxazole derivatives, a process for the preparation thereof, and radiation-sensitive compositions containing these derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1983-02-01 US disclosed
EP-0041675-A2 4-Halogen-5-(trichloromethyl-phenyl)-oxazole derivatives, process for preparing them and radiation-sensitive compositions containing them HOECHST AKTIENGESELLSCHAFT (DE) 1981-12-16 EP disclosed
US-4017313-A Photosensitive composition containing a leuco dye, a photosensitizer, an aromatic aldehyde and a secondary or tertiary amine and the use thereof in a direct-print process E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-04-12 US disclosed