SCHEMBL8716258

SCHEMBL8716258

COc1ccc(CC(C)(C[C@H](N)O)c2ccc(OC)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.44
CASR P41180 6/20 0.42
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
AOC3 Q16853 1/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
EPHX2 P34913 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
IDO1 P14902 1/20 0.39
AGXT P21549 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
LDHA P00338 1/20 0.38
KIF11 P52732 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716720 0.83 CASR (0.49) SLC6A4CASRNPC1RAB9AKMT2A
SCHEMBL8718475 0.78 MAOB (0.48) CYP1A2CYP2C19NPC1EPHX2RAB9A
SCHEMBL8720161 0.78 TAAR1 (0.48) CYP1A2AOC3IDO1AGXTTAAR1
SCHEMBL8714023 0.78 TRPA1 (0.46) SLC6A4ESR1ESR2CYP1A2CYP2D6
SCHEMBL8714103 0.77 EPHX2 (0.41) EPHX2LDHA
SCHEMBL8717242 0.77 ESR1 (0.46) SLC6A4ESR1ESR2LDHA
SCHEMBL8712989 0.76 MMP1 (0.43) KMT2A
SCHEMBL8716544 0.76 ESR1 (0.40) CASRESR1ESR2MEN1NPC1
SCHEMBL8716608 0.76 KIF11 (0.44) ESR1ESR2CYP1A2CYP2C19MEN1
SCHEMBL8713320 0.76 ESR1 (0.38) ESR1ESR2CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811293-A CULTURE PRODUCT AS CHEMICAL INTERMEDIATE FOR ANTI-OBESITY AGENT DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-22 US disclosed