SCHEMBL8716953

SCHEMBL8716953

O=C([C@H](O)c1ccccc1)N(CC1CCCNC1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.53
KMT2A Q03164 1/20 0.46
GHSR Q92847 6/20 0.43
CHRNB2 P17787 3/20 0.41
CHRNA4 P43681 3/20 0.41
CHRNB4 P30926 2/20 0.41
CHRNA3 P32297 2/20 0.41
ATM Q13315 1/20 0.38
USP30 Q70CQ3 1/20 0.38
CPN1 P15169 1/20 0.38
CPB2 Q96IY4 1/20 0.38
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 2/20 0.36
KCNH2 Q12809 1/20 0.36
CYP2D6 P10635 1/20 0.36
HTT P42858 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567800 0.79 GPR88 (0.55) GPR88KMT2ACHRNB2CHRNA4CHRNB4
Mandelic Acid SCHEMBL6950424 0.74 KMT2A (0.49) KMT2ACHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL3611085 0.71 GHSR (0.48) GPR88KMT2AGHSRCHRNB2CHRNA4
SCHEMBL9996441 0.71 GHSR (0.48) GPR88KMT2AGHSRCHRNB2CHRNA4
SCHEMBL14194158 0.71 OPRM1 (0.48) GPR88KMT2ACHRNB2CHRNA4CHRNB4
SCHEMBL10869689 0.70 KMT2A (0.53) GPR88KMT2ACHRNB2CHRNA4CHRNB4
Mandelic Acid SCHEMBL23121138 0.70 KMT2A (0.44) KMT2ACHRNB2CHRNA4CHRNB4CHRNA3
Mandelic Acid SCHEMBL7297870 0.70 KMT2A (0.50) KMT2A
Mandelic Acid SCHEMBL6974418 0.70 KMT2A (0.44) KMT2ACHRNB2CHRNA4CHRNB4CHRNA3
Mandelic Acid SCHEMBL8716945 0.70 KMT2A (0.50) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763604-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
US-5677448-A CHEMICAL INTERMEDIATES FOR MAKING ANTAGONIST OF THROMBIN, TREATING THROMBOSIS, STROKE, INFLAMMATION, ARTERIOSCLEROSIS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-10-14 US disclosed
US-5578594-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1996-11-26 US disclosed
US-5405854-A Anticoagulants HOFFMANN-LA ROCHE INC. (US) 1995-04-11 US disclosed