SCHEMBL8717074

SCHEMBL8717074

Fc1cc(C2CCCNC2)c2cn[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.43
HTR2C P28335 7/20 0.43
DRD2 P14416 1/20 0.43
KCNH2 Q12809 1/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
METAP2 P50579 1/20 0.40
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
JAK3 P52333 1/20 0.37
HTR2B P41595 2/20 0.37
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1E P28566 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37
TDO2 P48775 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7775075 0.78 HTR2A (0.43) HTR2AHTR2CDRD2KCNH2ROCK2
SCHEMBL8470311 0.77 METAP2 (0.40) ROCK2ROCK1METAP2TDO2
SCHEMBL24127329 0.69 DRD2 (0.47) HTR2AHTR2CDRD2KCNH2HTR2B
SCHEMBL22619200 0.69 NOS1 (0.44) METAP2
SCHEMBL17738576 0.67 JAK2 (0.51) METAP2JAK2JAK1TYK2JAK3
SCHEMBL2781869 0.66 SLC6A4 (0.56) HTR2AHTR2CDRD2KCNH2HTR2B
SCHEMBL30403358 0.65 METAP2 (0.56) METAP2TDO2
SCHEMBL3538351 0.65 METAP2 (0.56) METAP2TDO2
SCHEMBL14028515 0.65 IKBKB (0.58) ROCK2ROCK1
SCHEMBL23469324 0.64 HTR2A (0.48) HTR2AHTR2CDRD2KCNH2HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776963-A ANTIPSYCHOTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-07-07 US disclosed