SCHEMBL7775075

SCHEMBL7775075

c1cc(C2CCCNC2)c2cn[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
KCNH2 Q12809 1/20 0.43
NOS1 P29475 3/20 0.41
AXL P30530 1/20 0.41
MET P08581 1/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
PARP1 P09874 1/20 0.40
TRPV1 Q8NER1 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22619200 0.91 NOS1 (0.44) NOS1AXLMETTRPV1
SCHEMBL14102482 0.85 NOS1 (0.49) NOS1AXLMETTRPV1
Hydrochloric Acid SCHEMBL4683856 0.83 NOS1 (0.47) NOS1AXLMETTRPV1
SCHEMBL8717074 0.78 HTR2A (0.43) HTR2AHTR2CKCNH2ROCK2ROCK1
SCHEMBL10491761 0.77 JAK2 (0.46) HTR2AHTR2CKCNH2DRD2DRD3
Hydrochloric Acid SCHEMBL11136214 0.75 JAK2 (0.45) HTR2AHTR2CKCNH2DRD2DRD3
SCHEMBL5415511 0.75 CHRNB2 (0.49) ROCK2ROCK1
SCHEMBL9044788 0.74 MTNR1A (0.50) HTR2AHTR2CKCNH2DRD2DRD3
Trifluoroacetic Acid SCHEMBL4687032 0.73 TRPV1 (0.44) AXLTRPV1
SCHEMBL24365522 0.72 MEN1 (0.44) NOS1AXLMETPARP1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251907-B1 1-(aryloxyalkyl)-4-(heteroaryl) piperazines and related compounds useful as antipsychotics and analgesics AVENTIS PHARMACEUTICALS INC. 2001-06-26 US disclosed