SCHEMBL871839

SCHEMBL871839

O=C(Nc1ccc(/C=C/c2ccc(N(C(=O)c3ccsc3)C(=O)[C@@H]3CCCN3)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 2/20 0.39
SCN3A Q9NY46 3/20 0.38
SCN9A Q15858 2/20 0.38
PFKFB3 Q16875 5/20 0.35
PFKFB1 P16118 4/20 0.35
PFKFB2 O60825 3/20 0.35
DHODH Q02127 2/20 0.35
ULK1 O75385 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
SCN5A Q14524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845510 0.78 SCN3A (0.54) PSMB8SCN3ASCN9APFKFB3PFKFB1
SCHEMBL845438 0.76 RHOC (0.41)
Hydrochloric Acid SCHEMBL16741983 0.73 SCN3A (0.52) PSMB8SCN3ASCN9APFKFB3PFKFB1
Hydrochloric Acid SCHEMBL16741981 0.73 SCN3A (0.52) PSMB8SCN3ASCN9APFKFB3PFKFB1
SCHEMBL10119356 0.71 CA12 (0.47) PSMB8SCN3ASCN9ADHODHHDAC3
SCHEMBL8236871 0.70 SCN3A (0.48) PSMB8SCN3ASCN9APFKFB3PFKFB1
SCHEMBL845568 0.69 RHOC (0.36)
SCHEMBL449568 0.69 SCN3A (0.52) PSMB8SCN3ASCN9APFKFB3PFKFB1
SCHEMBL449567 0.69 SCN3A (0.52) PSMB8SCN3ASCN9APFKFB3PFKFB1
SCHEMBL845565 0.69 KMT2A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed