SCHEMBL8722147

SCHEMBL8722147

Cc1cc(C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc(C)c1Oc1ccc(N(CCBr)CCBr)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.39
CA1 P00915 2/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
TYMS P04818 1/20 0.38
KDR P35968 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
PRSS1 P07477 2/20 0.34
TMPRSS15 P98073 2/20 0.34
DHFR P00374 1/20 0.34
FOLH1 Q04609 1/20 0.34
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8722961 0.90 CA2 (0.46) CA2CA1CA12CA9TYMS
SCHEMBL8728048 0.86 CA1 (0.40) CA2CA1CA12CA9TAS1R3
SCHEMBL8726522 0.83 CA2 (0.46) CA2CA1CA12CA9TYMS
SCHEMBL8724180 0.82 CA2 (0.45) CA2CA1CA12CA9TYMS
SCHEMBL8726202 0.81 CA2 (0.46) CA2CA1CA12CA9TYMS
SCHEMBL8722076 0.81 CA2 (0.41) CA2CA1CA12CA9TYMS
SCHEMBL8724224 0.80 CA2 (0.46) CA2CA1CA12CA9TYMS
SCHEMBL8726160 0.79 MAPT (0.36) CA1CA12CA9TAS1R3TAS1R1
SCHEMBL8722941 0.79 CA2 (0.41) CA2CA1CA12CA9TYMS
SCHEMBL8722628 0.78 MMP2 (0.37) CA2CA1CA12CA9TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998035982-A1 COMPOUNDS FOR USE IN ADEPT ZENECA LIMITED (GB) 1998-08-20 WO disclosed