SCHEMBL8726160

SCHEMBL8726160

Cc1cc(C(=O)N[C@@H](C)C(=O)OC(C)(C)C)cc(C)c1Oc1ccc(N(CCBr)CCBr)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.36
NPSR1 Q6W5P4 5/20 0.36
TDP1 Q9NUW8 5/20 0.36
XBP1 P17861 3/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPK1 P28482 1/20 0.33
ATM Q13315 1/20 0.33
ALDH1A1 P00352 3/20 0.33
POLB P06746 1/20 0.33
RECQL P46063 3/20 0.33
GPR55 Q9Y2T6 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726452 0.88 MAPT (0.40) MAPTNPSR1TDP1XBP1KDM4E
SCHEMBL8728048 0.88 CA1 (0.40) TAS1R3TAS1R1KDM4EALDH1A1CA12
SCHEMBL8722057 0.81 HRH3 (0.41) MAPTNPSR1TDP1XBP1MAPK1
SCHEMBL8722967 0.80 ALDH1A1 (0.41) MAPTNPSR1TDP1XBP1MAPK1
SCHEMBL8722147 0.79 CA2 (0.39) TAS1R3TAS1R1KDM4ECA12CA1
SCHEMBL8727998 0.77 TAS1R3 (0.46) MAPTNPSR1TDP1XBP1TAS1R3
SCHEMBL8724198 0.77 TAS1R3 (0.37) MAPTNPSR1TAS1R3TAS1R1MAPK1
SCHEMBL8726226 0.76 CA1 (0.49) MAPTNPSR1KDM4EALDH1A1CA12
SCHEMBL8724211 0.72 MAPT (0.41) MAPTNPSR1TDP1XBP1MAPK1
SCHEMBL7717390 0.71 MAPT (0.36) MAPTNPSR1TDP1XBP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998035982-A1 COMPOUNDS FOR USE IN ADEPT ZENECA LIMITED (GB) 1998-08-20 WO disclosed