SCHEMBL8722264

SCHEMBL8722264

CN(CCC(Oc1ccc(C(F)(F)F)cc1)c1ccccc1)C(=O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 14/20 0.61
SLC6A4 P31645 3/20 0.59
HRH3 Q9Y5N1 2/20 0.59
HTR1A P08908 1/20 0.58
NPC1 O15118 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C19 P33261 2/20 0.48
MTOR P42345 2/20 0.48
RAB9A P51151 2/20 0.48
SLC6A2 P23975 2/20 0.48
SLC6A3 Q01959 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
ALOX15 P16050 1/20 0.48
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5269933 0.90 SLC6A9 (0.71) SLC6A9SLC6A4HRH3NPC1CYP2D6
SCHEMBL8726597 0.89 SLC6A9 (0.57) SLC6A9SLC6A4HRH3HTR1ANPC1
SCHEMBL7943023 0.85 SLC6A9 (0.72) SLC6A9SLC6A4HRH3NPC1CYP2D6
SCHEMBL8931276 0.84 SLC6A4 (0.64) SLC6A9SLC6A4HRH3HTR1ANPC1
SCHEMBL8726521 0.83 SLC6A9 (0.63) SLC6A9SLC6A4HRH3HTR1ANPC1
SCHEMBL13780465 0.81 SLC6A9 (0.77) SLC6A9SLC6A4HRH3NPC1CYP2D6
SCHEMBL7939788 0.81 SLC6A9 (0.69) SLC6A9SLC6A4HRH3NPC1CYP2D6
SCHEMBL8204423 0.80 SLC6A9 (0.60) SLC6A9SLC6A4HRH3NPC1CYP2D6
SCHEMBL8931267 0.79 ALDH1A1 (0.44) SLC6A9SLC6A4HTR1AACHE
SCHEMBL8722262 0.79 SLC6A9 (0.67) SLC6A9SLC6A4HRH3NPC1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0617006-B1 N-Substituted derivatives of N-methyl-3-(p-trifluoromethylphenoxy)-3-phenylpropylamine and procedure for their preparation PLIVA PHARM & CHEM WORKS (HR) 1998-05-06 EP disclosed
US-5618968-A N-substituted derivatives of N-methyl-3-(p-trifluoromethylphenoxy)-3-phenylpropylamine and the procedure for their preparation PLIVA FARMACEUTSKA KEMIJSKA, PREHRAMBENA I KOZMETICKA INDUSTRIJA, DIONICKO DRUSTVO (HR) 1997-04-08 US disclosed
EP-0617006-A1 N-subtituted derivatives of N-methyl-3-(p-trifluoromethylphenoxy)-3-phenylpropylamine and the procedure for their preparation PLIVA d.d. ZAGREB (HR) 1994-09-28 EP disclosed