SCHEMBL8723723

SCHEMBL8723723

[CH]c1cccc(C(Br)Br)c1

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 1/20 0.31
PGK2 P07205 1/20 0.31
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250314 0.81 PGK1 (0.42) PGK1PGK2CES2CES1TRPA1
SCHEMBL8723919 0.75 TSHR (0.48) PGK1PGK2
SCHEMBL642404 0.72 IDO1 (0.48)
SCHEMBL2186969 0.71
SCHEMBL7305650 0.70 PGK1 (0.35) PGK1PGK2CES2CES1TRPA1
SCHEMBL28420 0.70 SLC6A3 (0.37) PGK1PGK2CES2CES1TRPA1
SCHEMBL384041 0.70 ACP3 (0.46)
SCHEMBL7305656 0.70 LMNA (0.52)
SCHEMBL20902925 0.70 PGK1 (0.31) PGK1PGK2CES2CES1TRPA1
SCHEMBL321883 0.70 ACHE (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609058-B1 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO CO (JP) 1998-12-09 EP disclosed
US-5491167-A INHIBITORS OF CHOLESTEROL BIOSYNTHESIS SANKYO COMPANY, LIMITED (JP) 1996-02-13 US disclosed
EP-0609058-A2 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1994-08-03 EP disclosed