SCHEMBL8723863

SCHEMBL8723863

O=C(Nc1ccc2[nH]cc(C3=CCN4CCCCC4CC3)c2c1)Nc1ccc(F)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.41
MAPT P10636 3/20 0.40
POLB P06746 1/20 0.40
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
STING1 Q86WV6 1/20 0.37
HTR1D P28221 1/20 0.37
DRD2 P14416 2/20 0.36
HTR1A P08908 1/20 0.36
DRD4 P21917 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR7 P34969 1/20 0.36
DRD3 P35462 1/20 0.36
HTR2B P41595 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720598 0.91 NOS3 (0.42) SLC6A4MAPTPOLBNOS3NOS1
SCHEMBL8725966 0.85 HTR1F (0.46) MAPTHTR1DHTR1AHTR2AHTR2C
SCHEMBL8724218 0.85 NOS3 (0.41) SLC6A4MAPTPOLBNOS3NOS1
SCHEMBL7486116 0.83 SLC6A4 (0.63) SLC6A4NOS3NOS1
SCHEMBL8721895 0.81 MAPT (0.42) SLC6A4MAPTPOLBNOS3NOS1
SCHEMBL8382132 0.81 HTR1D (0.40) SLC6A4MAPTPOLBNOS3NOS1
SCHEMBL8385402 0.79 MAPT (0.41) MAPTPOLBNOS3NOS1STING1
SCHEMBL8387232 0.77 SLC6A4 (0.55) SLC6A4HTR1DDRD2HTR1A
SCHEMBL8721897 0.77 NOS3 (0.43) SLC6A4MAPTNOS3NOS1DRD2
SCHEMBL8383659 0.76 MAPT (0.43) SLC6A4MAPTNOS3NOS1STING1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0875513-A1 Substituted heteroaromatic 5-HT 1F agonists ELI LILLY AND COMPANY (US) 1998-11-04 EP disclosed