SCHEMBL872553

SCHEMBL872553

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)Cc3ccncc3)cc2)cc1)[C@@H]1C=CCN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
GLA P06280 1/20 0.35
HDAC1 Q13547 1/20 0.33
SMN1; SMN2 Q16637 5/20 0.32
LMNA P02545 4/20 0.32
POLB P06746 2/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HTT P42858 2/20 0.31
TSHR P16473 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
F10 P00742 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA5A P35218 1/20 0.30
CA7 P43166 1/20 0.30
CA5B Q9Y2D0 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845099 0.91 ITGB1 (0.44) ITGB1ITGA4GLAHDAC1SMN1; SMN2
SCHEMBL872288 0.90 ITGB1 (0.37) ITGB1ITGA4POLBPDE3BPARP1
SCHEMBL845098 0.87 ITGB1 (0.43) ITGB1ITGA4GLAHDAC1SMN1; SMN2
SCHEMBL10119279 0.85 EPHX2 (0.37) ITGB1ITGA4KMT2ACA1CA2
SCHEMBL13272184 0.83 PDE3B (0.34) ITGB1ITGA4KMT2APDE3BPDE3A
SCHEMBL845622 0.79 ITGB1 (0.42) ITGB1ITGA4POLBALDH1A1HTT
SCHEMBL872031 0.79 PTPN1 (0.34) SMN1; SMN2LMNAPOLBKMT2AALDH1A1
SCHEMBL845351 0.76 ITGB1 (0.41) ITGB1ITGA4POLBKMT2AALDH1A1
SCHEMBL845190 0.74 EPHX2 (0.42) ITGB1ITGA4KMT2ACA1CA2
SCHEMBL845214 0.74 ITGB1 (0.39) ITGB1ITGA4LMNAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed