SCHEMBL845351

SCHEMBL845351

CC(=O)N1CC=C[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)Cc3cccnc3)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
PAX8 Q06710 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
TBXAS1 P24557 2/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
CYP17A1 P05093 1/20 0.37
CYP21A2 P08686 1/20 0.37
CYP11B1 P15538 1/20 0.37
THRB P10828 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845622 0.96 ITGB1 (0.42) ITGB1ITGA4PAX8HRH3TBXAS1
SCHEMBL845334 0.89 ITGB1 (0.39) ITGB1ITGA4PAX8HRH3TBXAS1
SCHEMBL845098 0.89 ITGB1 (0.43) ITGB1ITGA4ALDH1A1HTTKMT2A
SCHEMBL872288 0.88 ITGB1 (0.37) ITGB1ITGA4PAX8HRH3TBXAS1
SCHEMBL873383 0.84 CHRNA7 (0.36) ALDH1A1HTTCYP17A1CYP21A2CYP11B1
SCHEMBL845099 0.84 ITGB1 (0.44) ITGB1ITGA4ALDH1A1HTTKMT2A
SCHEMBL845086 0.82 EPHX2 (0.40) ITGB1ITGA4ALDH1A1KMT2AMAPT
SCHEMBL845097 0.82 NAMPT (0.39) ITGB1ITGA4ALDH1A1HTTKMT2A
SCHEMBL845401 0.81 ALDH1A1 (0.45) ITGB1ITGA4PAX8HRH3ALDH1A1
SCHEMBL10119337 0.79 ADRB1 (0.36) ITGB1ITGA4PAX8HRH3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed