SCHEMBL872288

SCHEMBL872288

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)Cc3cccnc3)cc2)cc1)[C@@H]1C=CCN1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.37
ITGA4 P13612 1/20 0.37
PAX8 Q06710 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
TBXAS1 P24557 2/20 0.34
PDE3B Q13370 1/20 0.34
TNKS O95271 1/20 0.34
PARP1 P09874 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
PARP4 Q9UKK3 1/20 0.34
PARP3 Q9Y6F1 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
POLB P06746 1/20 0.33
NAMPT P43490 2/20 0.33
CLK2 P49760 1/20 0.33
CLK3 P49761 1/20 0.33
DYRK1A Q13627 1/20 0.33
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845622 0.91 ITGB1 (0.42) ITGB1ITGA4PAX8HRH3TBXAS1
SCHEMBL872553 0.90 ITGB1 (0.39) ITGB1ITGA4PDE3BPARP1POLB
SCHEMBL845351 0.88 ITGB1 (0.41) ITGB1ITGA4PAX8HRH3TBXAS1
SCHEMBL10119279 0.84 EPHX2 (0.37) ITGB1ITGA4PARP1HTR1ADRD2
SCHEMBL845334 0.84 ITGB1 (0.39) ITGB1ITGA4PAX8HRH3TBXAS1
SCHEMBL845099 0.80 ITGB1 (0.44) ITGB1ITGA4PDE3BPOLB
SCHEMBL13272184 0.80 PDE3B (0.34) ITGB1ITGA4PAX8PDE3BNAMPT
SCHEMBL872031 0.78 PTPN1 (0.34) POLBNAMPT
SCHEMBL845098 0.77 ITGB1 (0.43) ITGB1ITGA4PDE3BPOLB
SCHEMBL10119337 0.75 ADRB1 (0.36) ITGB1ITGA4PAX8HRH3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed